SCHEMBL20154316

SCHEMBL20154316

CCOC(=O)CC(NSC(C)(C)C)c1cnc2ccccc2n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
KDM4E B2RXH2 2/20 0.48
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
HIF1A Q16665 1/20 0.44
KMT2A Q03164 5/20 0.41
RAB9A P51151 5/20 0.41
MEN1 O00255 4/20 0.41
NPC1 O15118 4/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
PRNP P04156 3/20 0.38
MAPT P10636 2/20 0.38
ABCB1 P08183 1/20 0.38
HTT P42858 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
FGFR2 P21802 2/20 0.37
FGFR3 P22607 2/20 0.37
FGFR1 P11362 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142638 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL20141004 0.77 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL29903077 0.77 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL18522686 0.74 MAPT (0.41) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL23259455 0.71 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2KDM4EKMT2ARAB9A
SCHEMBL24307417 0.70 ALDH1A1 (0.40) ALDH1A1KDM4EMAPTHTTL3MBTL1
SCHEMBL12603197 0.69 SMN1; SMN2 (0.32) ALDH1A1SMN1; SMN2KDM4EKMT2AMEN1
SCHEMBL4651782 0.67 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL25412903 0.67 CYP1A2 (0.64) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL20154296 0.67 KDM4E (0.40) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089360-A1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed