SCHEMBL20154319

SCHEMBL20154319

CCOC(=O)C[C@H](NC(=O)c1cc(CCc2ccc3c(n2)NCCC3)c[nH]1)c1ccc(OC)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.53
ITGAV P06756 19/20 0.53
ITGB6 P18564 12/20 0.51
ITGB5 P18084 12/20 0.51
ITGB8 P26012 11/20 0.51
ITGA2B P08514 1/20 0.51
CXCR4 P61073 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21271427 0.92 ITGB3 (0.61) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL20154377 0.92 ITGB3 (0.61) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL29903058 0.92 ITGB3 (0.61) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21271503 0.92 ITGB3 (0.61) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21284325 0.85 ITGB3 (0.45) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21311505 0.82 ITGB3 (0.60) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21317575 0.81 ITGB3 (0.53) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL30487491 0.81 ITGB3 (0.53) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21271484 0.80 ITGB3 (0.61) ITGB3ITGAVITGB6ITGB5ITGB8
SCHEMBL21271488 0.80 ITGB3 (0.61) ITGB3ITGAVITGB6ITGB5ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538528-B1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2020-12-23 EP disclosed
WO-2018089360-A1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed