SCHEMBL20154948

SCHEMBL20154948

NC(=O)c1cc(Oc2ccc(F)cc2F)c(Br)cc1N

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.46
BRD4 O60885 4/20 0.44
PKM P14618 1/20 0.40
DGAT1 O75907 1/20 0.39
SCN4A P35499 1/20 0.39
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
HSPB1 P04792 2/20 0.37
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KEAP1 Q14145 1/20 0.36
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15067206 0.86 KDM4E (0.48) EPAS1BRD4PKMALDH1A1GAA
SCHEMBL30194335 0.82 EPAS1 (0.51) EPAS1PKMHSPB1ALDH1A1L3MBTL1
SCHEMBL16738742 0.82 EPAS1 (0.51) EPAS1PKMHSPB1ALDH1A1L3MBTL1
SCHEMBL20155384 0.81 HSPB1 (0.53) EPAS1BRD4LMNAHTTHSPB1
SCHEMBL16047284 0.81 EPAS1 (0.50) EPAS1PKMHSPB1ALDH1A1L3MBTL1
SCHEMBL16047925 0.81 EPAS1 (0.50) EPAS1PKMHSPB1ALDH1A1L3MBTL1
SCHEMBL2443815 0.79 EPAS1 (0.48) EPAS1BRD4HSPB1ALDH1A1
SCHEMBL4855967 0.78 HSPB1 (0.50) BRD4SCN4AHSPB1ALDH1A1KEAP1
SCHEMBL15067364 0.77 BRD4 (0.58) EPAS1BRD4ALDH1A1HPGD
SCHEMBL16048593 0.76 EPAS1 (0.48) EPAS1HSPB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed