SCHEMBL20155013

SCHEMBL20155013

CCS(=O)(=O)Cc1ccc(OCC2CC2)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.36
PDE4B Q07343 2/20 0.33
RORC P51449 9/20 0.33
PDE4A P27815 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
DUT P33316 1/20 0.32
IL17A Q16552 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21190849 0.90 BRD4 (0.44) BRD4PDE4BRORCPDE4APDE4C
SCHEMBL16658431 0.86 LPL (0.35) BRD4
SCHEMBL1438795 0.86 LPL (0.35) PDE4BRORCPDE4APDE4CPDE4D
SCHEMBL15069539 0.82 BRD4 (0.46) BRD4RORCPTGS1PTGS2
SCHEMBL16650807 0.81 BRD4 (0.44) BRD4
SCHEMBL984993 0.81 CNR2 (0.35) PDE4B
SCHEMBL16651855 0.81 BRD4 (0.47) BRD4PTGS1PTGS2
SCHEMBL21191141 0.81 BRD4 (0.39) BRD4PDE4BRORCPDE4APDE4C
SCHEMBL16650483 0.79 BRD4 (0.46) BRD4
SCHEMBL21190751 0.78 BRD4 (0.45) BRD4PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed