SCHEMBL20155028

SCHEMBL20155028

Cn1cc2c(=O)n(C)cc(-c3cc(N)ccc3Oc3ccc(Cl)cc3C#N)c2n1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.41
SCN9A Q15858 13/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155476 0.89 BRD4 (0.43) BRD4
SCHEMBL20155554 0.88 BRD4 (0.42) BRD4ALDH1A1GAA
SCHEMBL20155411 0.86 BRD4 (0.47) BRD4
SCHEMBL20155360 0.84 BRD4 (0.49) BRD4KDM4EALDH1A1
SCHEMBL20155020 0.84 BRD4 (0.42) BRD4SCN9A
SCHEMBL20155019 0.83 BRD4 (0.57) BRD4
SCHEMBL20155420 0.83 BRD4 (0.42) BRD4
SCHEMBL20155002 0.82 BRD4 (0.49) BRD4SCN9A
SCHEMBL20155478 0.81 BRD4 (0.43) BRD4
SCHEMBL20155702 0.81 BRD4 (0.40) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed