SCHEMBL20155071

SCHEMBL20155071

Cn1cc(Br)c2c(cc(CN3CCN(C(=O)OC(C)(C)C)CC3)n2COCC[Si](C)(C)C)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 3/20 0.37
PLK1 P53350 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
VEGFA P15692 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
DDR1 Q08345 2/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
IDO2 Q6ZQW0 1/20 0.34
KCNH2 Q12809 1/20 0.34
GPR119 Q8TDV5 2/20 0.34
P2RY14 Q15391 1/20 0.34
RET P07949 1/20 0.34
CHRM2 P08172 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20154954 0.97 PARP1 (0.37) ACKR3PLK1CA12CA1CA2
SCHEMBL20154962 0.86 NPC1 (0.33) DDR1NPC1
SCHEMBL20155261 0.83 SMN1; SMN2 (0.35) NPC1
SCHEMBL20155678 0.83 CHKA (0.33) NPC1
SCHEMBL20155070 0.78 BRD4 (0.45) PLK1IDO1TDO2IDO2
SCHEMBL20154958 0.78 NPC1 (0.39) NPC1
SCHEMBL26128638 0.78 CCNK (0.37) ACKR3VEGFAEGLN1KCNH2GPR119
SCHEMBL20154951 0.76 NPC1 (0.36) NPC1
SCHEMBL20155074 0.75 BRD4 (0.51)
SCHEMBL20154956 0.73 BRD4 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed