SCHEMBL20154962

SCHEMBL20154962

CN1CCN(Cc2cc3c(=O)n(C)cc(Br)c3n2COCC[Si](C)(C)C)CC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
KDM4E B2RXH2 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TSHR P16473 1/20 0.32
ALDH1A1 P00352 3/20 0.31
PIM1 P11309 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
HTR1B P28222 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DGAT1 O75907 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155678 0.96 CHKA (0.33) NPC1KDM4ETDP1SMN1; SMN2TSHR
SCHEMBL20155261 0.91 SMN1; SMN2 (0.35) NPC1KDM4ESMN1; SMN2ALDH1A1GAA
SCHEMBL20155071 0.86 ACKR3 (0.37) NPC1DDR1
SCHEMBL20154958 0.83 NPC1 (0.39) NPC1DGAT1
SCHEMBL20154951 0.83 NPC1 (0.36) NPC1DGAT1
SCHEMBL20154954 0.83 PARP1 (0.37) KMT2ADDR1
SCHEMBL20155035 0.77 NPC1 (0.36) NPC1DGAT1
SCHEMBL20155034 0.76 NPC1 (0.36) NPC1DGAT1
SCHEMBL20154955 0.76 KDM4C (0.32) NPC1
SCHEMBL31440547 0.75 NPC1 (0.39) NPC1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed