SCHEMBL20155488

SCHEMBL20155488

CCOn1cc2c(=O)[nH]ccc2n1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 1/20 0.38
PRKACA P17612 1/20 0.32
PRKACG P22612 1/20 0.32
PRKACB P22694 1/20 0.32
PARP1 P09874 1/20 0.32
JAK2 O60674 2/20 0.31
ELANE P08246 1/20 0.31
ATM Q13315 1/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
BLM P54132 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155518 0.83 KDM4E (0.36) KDM4EALDH1A1HPGDNPSR1PRKACA
SCHEMBL20155602 0.80 IP6K1 (0.40) KDM4EALDH1A1HPGDPARP1JAK2
SCHEMBL20155622 0.79 JAK2 (0.34) KDM4EALDH1A1HPGDNPSR1PARP1
SCHEMBL22216158 0.74 PARP1 (0.37) KDM4EALDH1A1HPGDNPSR1PARP1
SCHEMBL20155157 0.72 GSK3B (0.30)
SCHEMBL20155613 0.70 PARP1 (0.38) KDM4EALDH1A1HPGDNPSR1PARP1
SCHEMBL24035859 0.70 PARP1 (0.34) KDM4EALDH1A1HPGDNPSR1PARP1
SCHEMBL20155606 0.68 ATM (0.36) ATMPOLBTHRB
SCHEMBL20155563 0.68 CNR2 (0.42) KDM4EALDH1A1HPGDJAK2
SCHEMBL22206944 0.67 CCNK (0.45) ALDH1A1MEN1GAAMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed