SCHEMBL20155644

SCHEMBL20155644

Cn1cc2c(=O)n(C)cc(-c3cc(N)c(F)cc3Nc3ccc(F)cc3F)c2n1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 16/20 0.45
MAPK14 Q16539 1/20 0.37
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155651 0.91 BRD4 (0.43) BRD4MAPK14TSHRHSD17B10MAPT
SCHEMBL20155427 0.89 BRD4 (0.48) BRD4MAPK14TSHRHSD17B10
SCHEMBL20155103 0.84 BRD4 (0.42) BRD4MAPK14TSHRHSD17B10MAPT
SCHEMBL20155634 0.80 BRD4 (0.48) BRD4TSHRHSD17B10
SCHEMBL20155122 0.80 BRD4 (0.51) BRD4
SCHEMBL20155185 0.80 BRD4 (0.42) BRD4TP53POLB
SCHEMBL20155619 0.80 BRD4 (0.46) BRD4
SCHEMBL20155426 0.79 BRD4 (0.51) BRD4
SCHEMBL20155737 0.79 BRD4 (0.47) BRD4
SCHEMBL20155168 0.79 BRD4 (0.40) BRD4MAPK14TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed