SCHEMBL20156253

SCHEMBL20156253

COC(=O)/C(=C/NCCc1ccc2c(n1)NCCC2)N=N

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 6/20 0.51
ITGAV P06756 14/20 0.47
ITGB3 P05106 12/20 0.47
ITGB6 P18564 8/20 0.44
ITGB5 P18084 6/20 0.43
ITGB8 P26012 3/20 0.43
ITGB1 P05556 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156247 0.89 ITGAV (0.52) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156319 0.82 CXCR4 (0.51) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156358 0.81 CXCR4 (0.52) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156009 0.79 CXCR4 (0.47) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156008 0.78 ITGAV (0.53) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156245 0.77 ITGAV (0.54) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156094 0.77 ITGAV (0.49) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156097 0.76 ITGAV (0.48) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL20156098 0.76 CXCR4 (0.47) CXCR4ITGAVITGB3ITGB6ITGB5
SCHEMBL26032494 0.76 ITGAV (0.54) CXCR4ITGAVITGB3ITGB6ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed