SCHEMBL20156094

SCHEMBL20156094

N=C/C(=C\NCCc1ccc2c(n1)NCCC2)C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 14/20 0.49
ITGB3 P05106 12/20 0.49
CXCR4 P61073 6/20 0.48
ITGB6 P18564 3/20 0.42
ITGB5 P18084 1/20 0.42
ITGB8 P26012 1/20 0.42
ITGA2B P08514 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156008 0.91 ITGAV (0.53) ITGAVITGB3CXCR4ITGB6ITGB5
SCHEMBL20156009 0.85 CXCR4 (0.47) ITGAVITGB3CXCR4ITGB6ITGB5
SCHEMBL20156245 0.84 ITGAV (0.54) ITGAVITGB3CXCR4ITGB6ITGB5
SCHEMBL20156054 0.83 ITGAV (0.47) ITGAVITGB3CXCR4ITGB6ITGA2B
SCHEMBL20156055 0.83 ITGAV (0.47) ITGAVITGB3CXCR4ITGB6ITGA2B
SCHEMBL20156097 0.83 ITGAV (0.48) ITGAVITGB3CXCR4ITGB6ITGB5
SCHEMBL20156256 0.82 ITGB3 (0.52) ITGAVITGB3CXCR4ITGB6ITGB5
SCHEMBL20156247 0.79 ITGAV (0.52) ITGAVITGB3CXCR4ITGB6ITGB5
SCHEMBL20156248 0.79 ITGAV (0.44) ITGAVITGB3CXCR4ITGB6
SCHEMBL23912918 0.79 ITGB3 (0.56) ITGAVITGB3CXCR4ITGB6ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538527-B1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2021-10-13 EP disclosed
WO-2018089358-A1 AZOLE AMIDES AND AMINES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed