SCHEMBL20156870

SCHEMBL20156870

C=Cc1cc(C(=O)OC)c(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
CA14 Q9ULX7 2/20 0.36
PDK2 Q15119 1/20 0.36
PDK4 Q16654 1/20 0.36
ERN1 O75460 1/20 0.35
KDM4E B2RXH2 4/20 0.35
GAA P10253 3/20 0.35
LMNA P02545 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
POLB P06746 1/20 0.35
NFKB1 P19838 1/20 0.35
XDH P47989 1/20 0.35
GFER P55789 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
FUT7 Q11130 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17262480 0.87 CYP3A4 (0.37) CA12CA1CA2CA7CA9
SCHEMBL27214492 0.85 GAA (0.39) GAALMNAPOLBALPLTSHR
SCHEMBL25774061 0.85 KDM4E (0.42) CA12CA1CA2CA7CA9
SCHEMBL10290728 0.85 CYP3A4 (0.38) CA12CA1CA2CA7CA9
SCHEMBL26122042 0.84 ERN1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL31306166 0.82 CA12 (0.38) CA12CA1CA2CA7CA9
SCHEMBL22802075 0.81 CA12 (0.42) CA12CA1CA2CA7CA9
SCHEMBL410165 0.79 ALPL (0.45) CA12CA1CA2CA7CA9
SCHEMBL522786 0.79 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL29296039 0.79 ERN1 (0.47) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192989-A2 PHTHALAZINONE COMPOUNDS AS PARP7 INHIBITORS AZKARRA THERAPEUTICS, INC. (US) 2023-10-05 WO disclosed
WO-2023192989-A2 PHTHALAZINONE COMPOUNDS AS PARP7 INHIBITORS AZKARRA THERAPEUTICS, INC. (US) 2023-10-05 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed