SCHEMBL20157348

SCHEMBL20157348

CCS(=O)(=O)Cc1ccc(C(=O)c2ccc(C)cc2)c(-c2cn(C)c(=O)cc2CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC10 Q969S8 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
BRD4 O60885 2/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KCNA5 P22460 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
BRD9 Q9H8M2 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
BAZ2A Q9UIF9 1/20 0.31
HDAC1 Q13547 1/20 0.31
NAMPT P43490 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157755 0.93 BRD4 (0.35) HDAC10HDAC6BRD4RAF1BRAF
SCHEMBL20157351 0.93 HDAC10 (0.36) HDAC10HDAC6PPARGPPARABRD4
SCHEMBL21362694 0.90 BRD4 (0.34) HDAC10HDAC6BRD4RAF1BRAF
SCHEMBL21550010 0.88 BRD4 (0.36) HDAC10HDAC6BRD4RAF1BRAF
SCHEMBL21564878 0.88 BRD4 (0.34) HDAC10HDAC6BRD4RAF1BRAF
SCHEMBL21362110 0.87 BRD4 (0.34) HDAC10HDAC6BRD4
SCHEMBL20158068 0.87 CREBBP (0.34) RAF1BRAFKCNA5KMT2AMEN1
SCHEMBL20157896 0.86 BRD4 (0.35) HDAC10HDAC6BRD4RAF1BRAF
SCHEMBL21564924 0.86 HDAC10 (0.36) HDAC10HDAC6BRD4PDCD1CD274
SCHEMBL21550125 0.86 ALDH1A1 (0.36) HDAC10HDAC6BRD4KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed