SCHEMBL20158010

SCHEMBL20158010

CCCCSNC(CC)c1cc(=O)n(C)cc1-c1cc(N)c(F)cc1C(=O)c1ccc(F)cc1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.32
RXFP1 Q9HBX9 2/20 0.31
MAPT P10636 2/20 0.31
MAPK14 Q16539 1/20 0.31
TP53 P04637 1/20 0.31
FAAH O00519 2/20 0.31
CNR2 P34972 1/20 0.31
THRB P10828 1/20 0.31
PRNP P04156 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362618 0.86 BRD4 (0.35) BRD4RXFP1MAPTMAPK14TP53
SCHEMBL21352162 0.78 BRD4 (0.32) BRD4MAPK14
SCHEMBL21362087 0.73 BRD4 (0.32) BRD4MAPK14
SCHEMBL21362208 0.72 BRD4 (0.36) BRD4
SCHEMBL21362620 0.71 BRD4 (0.38) BRD4
SCHEMBL21362086 0.71 BRD4 (0.34) BRD4MAPK14CNR2
SCHEMBL20158149 0.70 GRM5 (0.33) BRD4MAPTMAPK14TP53
SCHEMBL21352227 0.70 BRD4 (0.32) BRD4MAPK14
SCHEMBL21351950 0.70 BRD4 (0.35) BRD4MAPTMAPK14THRB
SCHEMBL21352234 0.69 BRD4 (0.32) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed