SCHEMBL21362618

SCHEMBL21362618

CCC(NS)c1cc(=O)n(C)cc1-c1cc(N)c(F)cc1C(=O)c1ccc(F)cc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.35
MAPT P10636 3/20 0.33
RXFP1 Q9HBX9 2/20 0.33
TP53 P04637 1/20 0.33
PRNP P04156 1/20 0.33
POLB P06746 1/20 0.33
MAP2K2 P36507 1/20 0.32
MAP2K1 Q02750 1/20 0.32
MAPK14 Q16539 1/20 0.32
ATM Q13315 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158010 0.86 BRD4 (0.32) BRD4MAPTRXFP1TP53PRNP
SCHEMBL20158149 0.80 GRM5 (0.33) BRD4MAPTTP53POLBMAP2K2
SCHEMBL21362620 0.79 BRD4 (0.38) BRD4
SCHEMBL21352162 0.79 BRD4 (0.32) BRD4MAP2K2MAP2K1MAPK14ATM
SCHEMBL21362087 0.78 BRD4 (0.32) BRD4MAPK14ATM
SCHEMBL20157715 0.76 BRD4 (0.33) BRD4MAPTRXFP1TP53ATM
SCHEMBL20157669 0.76 BRD4 (0.37) BRD4
SCHEMBL21362208 0.75 BRD4 (0.36) BRD4
SCHEMBL21362239 0.72 BRD4 (0.42) BRD4
SCHEMBL21354531 0.72 BRD4 (0.31) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed