SCHEMBL20159155

SCHEMBL20159155

Cc1cccc(N2CCN(C(=O)c3cc(CN4CCN(c5ccccc5C#N)CC4)c(C)n3C)CC2)n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 6/20 0.65
RPTOR Q8N122 6/20 0.65
MLST8 Q9BVC4 6/20 0.65
DRD3 P35462 5/20 0.42
DRD4 P21917 3/20 0.42
DRD2 P14416 3/20 0.42
HTR2A P28223 3/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
THPO P40225 1/20 0.42
HIF1A Q16665 1/20 0.42
HTR1A P08908 3/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
NPC1 O15118 1/20 0.41
TACR3 P29371 1/20 0.41
PHGDH O43175 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159230 0.92 MTOR (0.65) MTORRPTORMLST8DRD3DRD4
SCHEMBL20159082 0.90 MTOR (0.75) MTORRPTORMLST8DRD3DRD4
SCHEMBL20158990 0.89 MTOR (0.77) MTORRPTORMLST8KDM4EALDH1A1
SCHEMBL20159131 0.87 MTOR (0.65) MTORRPTORMLST8DRD3DRD4
SCHEMBL20159229 0.86 MTOR (0.74) MTORRPTORMLST8DRD3DRD2
SCHEMBL20159090 0.86 MTOR (0.71) MTORRPTORMLST8DRD3DRD4
SCHEMBL20158992 0.86 MTOR (0.84) MTORRPTORMLST8DRD3DRD4
SCHEMBL20159152 0.85 MTOR (0.65) MTORRPTORMLST8DRD3DRD4
SCHEMBL20159156 0.85 MTOR (0.64) MTORRPTORMLST8DRD3DRD4
SCHEMBL20159153 0.84 MTOR (0.61) MTORRPTORMLST8DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed