SCHEMBL20159650

SCHEMBL20159650

CC(C)n1nc(N)nc1Oc1cccc(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 4/20 0.51
PSEN2 P49810 4/20 0.51
APH1B Q8WW43 4/20 0.51
NCSTN Q92542 4/20 0.51
APH1A Q96BI3 4/20 0.51
PSENEN Q9NZ42 4/20 0.51
HTR1A P08908 2/20 0.41
DRD2 P14416 2/20 0.41
HTR7 P34969 2/20 0.41
HTR6 P50406 2/20 0.41
HTR2A P28223 1/20 0.41
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
MAP4K4 O95819 1/20 0.39
OGG1 O15527 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
SRC P12931 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138690 0.84 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20159730 0.84 MAP4K4 (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL20159299 0.74 HTR2A (0.37) HTR2ASRCABL1MGLL
SCHEMBL23492813 0.71 PSEN1 (0.68) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL23492814 0.71 PSEN1 (0.68) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL23492815 0.71 PSEN1 (0.68) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL19361349 0.69 ABL1 (0.59) SRCABL1
SCHEMBL5556169 0.69 CYP1A2 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5560726 0.69 CYP1A2 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9369867 0.68 MEN1 (0.69) CYP1A2CYP2C9CYP2C19MAP4K4SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed