SCHEMBL20159709

SCHEMBL20159709

CCC1CC(=O)N(C)N=C1c1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.40
PDE2A O00408 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
ADORA2B P29275 2/20 0.34
ADORA1 P30542 1/20 0.34
MAOA P21397 1/20 0.34
CES2 O00748 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138813 0.81 PDE4A (0.40) CYP19A1PDE3BPDE3AKDM4EMEN1
SCHEMBL20142927 0.81 PDE4A (0.40) CYP19A1PDE3BPDE3AKDM4EMEN1
SCHEMBL20159190 0.81 PDE4A (0.40) CYP19A1PDE3BPDE3AKDM4EMEN1
SCHEMBL20159106 0.77 HRH3 (0.38) CYP19A1CES2KDM4EMEN1ALDH1A1
SCHEMBL20159497 0.75 CYP19A1 (0.48) CYP19A1CES2KDM4EMEN1ALDH1A1
SCHEMBL6655180 0.75 PDE4B (0.44)
SCHEMBL6842079 0.72 PDE4B (0.52) CYP19A1
SCHEMBL20142921 0.71 PDE4B (0.40) CYP19A1PDE3BPDE3ACES2KDM4E
SCHEMBL6654160 0.71 PDE4D (0.52) PDE3BPDE3A
SCHEMBL6684566 0.69 PDE4D (0.48) PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed