SCHEMBL20159902

SCHEMBL20159902

Cc1nnc2c(N)cc(-c3cc4[nH]ncc4cc3Oc3ccc(F)cc3F)nn12

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.38
TRPA1 O75762 2/20 0.35
BRD4 O60885 7/20 0.34
BTK Q06187 2/20 0.33
FYN P06241 1/20 0.33
SRC P12931 1/20 0.33
TEC P42680 1/20 0.33
ITK Q08881 1/20 0.33
ROCK2 O75116 1/20 0.33
TLR8 Q9NR97 1/20 0.33
ROCK1 Q13464 1/20 0.32
MAPK8 P45983 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159885 0.86 BRD4 (0.36) MAPK14BRD4MAPK8
SCHEMBL20160229 0.75 BRD4 (0.44) MAPK14TRPA1BRD4
SCHEMBL20155327 0.74 TRPA1 (0.45) MAPK14TRPA1BRD4TLR8MAPK8
SCHEMBL20159872 0.73 BRD4 (0.51) BRD4
SCHEMBL20160050 0.72 BRD4 (0.46) MAPK14BRD4
SCHEMBL20160251 0.71 BRD4 (0.41) BRD4
SCHEMBL20160026 0.70 BRD4 (0.42) MAPK14BRD4
SCHEMBL20160240 0.70 BRD4 (0.49) MAPK14BRD4MAPK8
SCHEMBL20160266 0.69 BRD4 (0.39) MAPK14TRPA1BRD4
SCHEMBL20160306 0.69 BRD4 (0.41) MAPK14BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed