SCHEMBL20159911

SCHEMBL20159911

Cc1cc(-c2cc(N)ccc2Oc2ccc(F)cc2F)cn2c(C)nnc12

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 17/20 0.43
BRD3 Q15059 7/20 0.36
BRD2 P25440 6/20 0.36
CREBBP Q92793 5/20 0.35
TRPA1 O75762 1/20 0.35
MAPK14 Q16539 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160236 0.93 BRD4 (0.43) BRD4BRD3BRD2TRPA1MAPK14
SCHEMBL20160322 0.85 BRD4 (0.39) BRD4BRD3BRD2
SCHEMBL20160241 0.84 PIM1 (0.44) BRD4MAPK14
SCHEMBL20160270 0.82 BRD4 (0.42) BRD4BRD3BRD2
SCHEMBL18538407 0.81 BRD4 (0.55) BRD4BRD3BRD2
SCHEMBL20160087 0.81 BRD4 (0.40) BRD4BRD2CREBBP
SCHEMBL20160232 0.81 BRD4 (0.39) BRD4BRD3BRD2
SCHEMBL20160233 0.80 BRD4 (0.55) BRD4BRD3BRD2
SCHEMBL20160229 0.79 BRD4 (0.44) BRD4TRPA1MAPK14
SCHEMBL20160253 0.77 BRD4 (0.38) BRD4MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed