SCHEMBL20159912

SCHEMBL20159912

Nc1cc(Cl)nn2cnnc12

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
HTT P42858 2/20 0.43
MAPT P10636 1/20 0.43
LMNA P02545 1/20 0.41
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 4/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.32
ADORA2A P29274 2/20 0.30
HAVCR2 Q8TDQ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31201339 0.80 KDM4E (0.47) KDM4EHTTMAPTLMNAALDH1A1
SCHEMBL21383755 0.73 KDM4E (0.49) KDM4EHTTMAPTLMNAALDH1A1
SCHEMBL5061012 0.73 KDM4E (0.41) KDM4EHTTMAPTLMNAALDH1A1
SCHEMBL31201372 0.73 KDM4E (0.43) KDM4EHTTMAPTLMNAALDH1A1
SCHEMBL23993919 0.73 KDM4E (0.43) KDM4EHTTMAPTLMNAALDH1A1
SCHEMBL2995450 0.69 SMPD3 (0.39) TDP1
SCHEMBL140145 0.68 KDM4E (0.39) KDM4EHTTMAPTLMNATDP1
SCHEMBL5061041 0.67 KDM4E (0.38) KDM4EHTTMAPTLMNAALDH1A1
SCHEMBL31201312 0.65 KDM4E (0.45) KDM4EHTTMAPTALDH1A1HPGD
SCHEMBL105123 0.65 BAZ2B (0.41) KDM4EHTTMAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4727944-A1 [1,2,4]-TRIAZOLO[4,3-B]PYRIDAZINE DERIVATIVES USEFUL AS A MEDICAMENT Perha Pharmaceuticals (FR) 2026-04-22 EP disclosed
US-20250275965-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS GRITSCIENCE BIOPHARMACEUTICALS CO LTD (CN) 2025-09-04 US disclosed
WO-2025080788-A1 CCR4 INHIBITORS AND METHODS OF USE THEREOF RAYTHERA, INC. (US) 2025-04-17 WO disclosed
WO-2024256496-A1 [1,2,4]-TRIAZOLO[4,3-B]PYRIDAZINE DERIVATIVES USEFUL AS A MEDICAMENT PERHA PHARMACEUTICALS (FR) 2024-12-19 WO disclosed
EP-4477653-A1 [1,2,4]-TRIAZOLO[4,3-B]PYRIDAZINE DERIVATIVES USEFUL AS A MEDICAMENT Perha Pharmaceuticals (FR) 2024-12-18 EP disclosed
CN-116888126-A Compound of casein kinase inhibitor 北京原基华毅生物科技有限公司 2023-10-13 CN disclosed
WO-2022127755-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2022-06-23 WO disclosed
WO-2022127755-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2022-06-23 WO disclosed
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250275965-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS PACSIN2, CSNK1A1, CSNK1G3 KDM4E 1702/4885HTT 3664/4885MAPT 489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.