SCHEMBL20160024

SCHEMBL20160024

Cc1nnc2ccc(-c3cc(N)ccc3Oc3ccc(F)cc3F)nn12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.45
L3MBTL1 Q9Y468 1/20 0.41
DPP4 P27487 1/20 0.38
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GABRA1 P14867 1/20 0.38
HPGD P15428 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPK14 Q16539 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160308 0.87 BRD4 (0.43) BRD4MAPK14KMT2ATRPA1
SCHEMBL20159887 0.85 BRD4 (0.41) BRD4L3MBTL1DPP4
SCHEMBL20160230 0.84 BRD4 (0.48) BRD4DPP4MAPK14TRPA1
SCHEMBL20160229 0.84 BRD4 (0.44) BRD4MAPK14TRPA1
SCHEMBL20160050 0.81 BRD4 (0.46) BRD4MAPK14
SCHEMBL20160251 0.80 BRD4 (0.41) BRD4
SCHEMBL20160273 0.80 SMN1; SMN2 (0.56) BRD4L3MBTL1KDM4ESMN1; SMN2
SCHEMBL20160293 0.79 BRD4 (0.43) BRD4KDM4ETDP1MAPK14SMN1; SMN2
SCHEMBL20160026 0.79 BRD4 (0.42) BRD4MAPK14
SCHEMBL20160241 0.78 PIM1 (0.44) BRD4MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed