SCHEMBL20160293

SCHEMBL20160293

Nc1ccc(Oc2ccc(F)cc2F)c(-c2ccc3nncn3n2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.43
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.36
MAPK14 Q16539 2/20 0.35
GAA P10253 1/20 0.34
SCN4A P35499 1/20 0.34
KDM4E B2RXH2 3/20 0.33
PSMD14 O00487 1/20 0.33
USP2 O75604 1/20 0.33
PRNP P04156 1/20 0.33
POLB P06746 1/20 0.33
MMP2 P08253 1/20 0.33
PTPN7 P35236 1/20 0.33
PPARG P37231 1/20 0.33
RECQL P46063 1/20 0.33
PPP1CA P62136 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
PTPN22 Q9Y2R2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159984 0.89 SMN1; SMN2 (0.35) BRD4NPC1HTTSMN1; SMN2GAA
SCHEMBL20160417 0.81 BRD4 (0.42) BRD4NPC1HTTSMN1; SMN2KDM4E
SCHEMBL20160024 0.79 BRD4 (0.45) BRD4SMN1; SMN2MAPK14KDM4EKMT2A
SCHEMBL20159904 0.78 MAPK14 (0.41) BRD4MAPK14SCN4A
SCHEMBL20160308 0.78 BRD4 (0.43) BRD4MAPK14KMT2A
SCHEMBL20159910 0.72 NPC1 (0.39) BRD4NPC1LMNA
SCHEMBL20160229 0.70 BRD4 (0.44) BRD4MAPK14SCN4A
SCHEMBL20160241 0.68 PIM1 (0.44) BRD4MAPK14
SCHEMBL20160230 0.67 BRD4 (0.48) BRD4MAPK14
SCHEMBL11628077 0.67 KDM4E (0.46) NPC1HTTSMN1; SMN2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed