SCHEMBL20160085

SCHEMBL20160085

COc1nnc2ccc(Br)nn12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 1/20 0.41
BRD4 O60885 7/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.32
LRRK2 Q5S007 1/20 0.31
PIM1 P11309 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MET P08581 1/20 0.31
CCL2 P13500 1/20 0.31
TAF1 P21675 1/20 0.31
BRD2 P25440 1/20 0.31
BRD3 Q15059 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17477291 0.78 KDM4E (0.58) KDM4EHPGDHSD17B10BRD4MEN1
SCHEMBL20160225 0.75 SMN1; SMN2 (0.51) KDM4EHPGDHSD17B10BRD4MEN1
SCHEMBL4817342 0.70 MAP4K4 (0.38) KDM4EHPGDHSD17B10MEN1KMT2A
SCHEMBL38661026 0.67 PIK3CA (0.41) KDM4EALDH1A1LMNAMAPTTSHR
SCHEMBL10490635 0.64 KDM4E (0.63) KDM4EHPGDHSD17B10BRD4ALDH1A1
SCHEMBL2763151 0.63 KDM4E (0.59) KDM4EHPGDHSD17B10MEN1KMT2A
SCHEMBL10764328 0.63 KDM4E (0.57) KDM4EHPGDHSD17B10BRD4MEN1
SCHEMBL9642720 0.59 LMNA (0.33) LMNASMN1; SMN2
SCHEMBL20160357 0.59 SCN5A (0.36)
SCHEMBL38664202 0.59 SCN5A (0.36) KDM4EHPGDHSD17B10ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086585-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed