SCHEMBL20160669

SCHEMBL20160669

CC(C)c1ccc(CN2CCN(C)C(=O)C2)nc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.50
PRMT5 O14744 3/20 0.44
WDR77 Q9BQA1 3/20 0.44
HRH3 Q9Y5N1 4/20 0.36
MDM2 Q00987 1/20 0.35
SLC2A1 P11166 1/20 0.35
SYK P43405 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
IDH1 O75874 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
DGKZ Q13574 1/20 0.33
SLC8A1 P32418 1/20 0.33
ENPP2 Q13822 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4293256 0.81 PIK3CD (0.45) PIK3CDPRMT5WDR77HRH3MDM2
SCHEMBL20160951 0.81 PIK3CD (0.45) PIK3CDPRMT5WDR77HRH3MDM2
SCHEMBL14924103 0.80 PRMT5 (0.44) PRMT5WDR77HRH3KDM4ELMNA
SCHEMBL12880866 0.77 HRH3 (0.51) PRMT5WDR77HRH3SYKALDH1A1
SCHEMBL13466409 0.77 HRH3 (0.48) PRMT5WDR77HRH3SYKHTT
SCHEMBL13466407 0.77 ALDH1A1 (0.49) PRMT5WDR77HRH3ALDH1A1KDM4E
SCHEMBL12880864 0.76 HRH3 (0.53) PRMT5WDR77HRH3HTTSMN1; SMN2
SCHEMBL19105585 0.74 PIM1 (0.46)
SCHEMBL20804006 0.74 IDH1 (0.38) PRMT5WDR77HRH3MDM2IDH1
SCHEMBL12028960 0.73 HRH3 (0.54) PRMT5WDR77HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086589-A1 1,5,7-TRI-SUBSTITUTED ISOQUINOLINE DERIVATIVES, PREPARATION THEREOF, AND USE THEREOF IN MEDICINES 上海海雁医药科技有限公司 2018-05-17 WO disclosed