SCHEMBL2016600

SCHEMBL2016600

CCOS(=O)(=O)Cc1cc(C#N)c2cccnc2c1-c1cccc(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.37
SCN9A Q15858 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
POLB P06746 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
TTK P33981 1/20 0.34
MAPK8 P45983 1/20 0.34
NLRP3 Q96P20 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.33
PIK3CD O00329 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018305 0.83 SCN9A (0.36) MAP4K4SCN9ANR1H2NR1H3PIK3CD
SCHEMBL2010638 0.78 MAP4K4 (0.40) MAP4K4KDM4EPIK3CDPDE4APDE4B
SCHEMBL2013332 0.78 MAP4K4 (0.42) MAP4K4KDM4EPIK3CDPDE4APDE4B
SCHEMBL2018303 0.74 PIK3CD (0.41) MAP4K4SCN9ANR1H2NR1H3PIK3CD
SCHEMBL2013344 0.73 MAP4K4 (0.41) MAP4K4KDM4EABCG2PIK3CDPDE4A
SCHEMBL2013331 0.72 PIK3CD (0.44) MAP4K4PIK3CDBCL2
SCHEMBL2010635 0.72 PIK3CD (0.44) MAP4K4PIK3CDPDE4APDE4BPDE4C
SCHEMBL2041671 0.71 ACLY (0.36) SCN9A
SCHEMBL12470338 0.70 PIK3CD (0.42) MAP4K4PIK3CDPDE4APDE4BPDE4C
SCHEMBL15621512 0.69 PIK3CD (0.43) MAP4K4PIK3CDBCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed