SCHEMBL20169314

SCHEMBL20169314

CS(C)(C)CCOCn1cc(C(F)(F)F)nc1-c1ccc(-c2ccc(O)nc2)cn1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.49
PTGS2 P35354 8/20 0.37
PTGS1 P23219 4/20 0.36
SDHB P21912 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
PMP22 Q01453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20169312 0.93 DGAT1 (0.53) DGAT1PTGS2PTGS1
SCHEMBL20169389 0.87 DGAT1 (0.47) DGAT1PTGS2PTGS1
SCHEMBL15293782 0.87 DGAT1 (0.66) DGAT1PTGS2
SCHEMBL20169313 0.86 DGAT1 (0.54) DGAT1PTGS2PTGS1
SCHEMBL20169340 0.86 DGAT1 (0.50) DGAT1PTGS2PTGS1
SCHEMBL20169318 0.85 DGAT1 (0.52) DGAT1PTGS2PTGS1KDM4EALDH1A1
SCHEMBL10176678 0.85 DGAT1 (0.47) DGAT1PTGS2PTGS1
SCHEMBL20169384 0.81 DGAT1 (0.49) DGAT1PTGS2PTGS1SDHBALDH1A1
SCHEMBL20169333 0.80 DGAT1 (0.74) DGAT1PTGS2PTGS1
SCHEMBL15293778 0.80 DGAT1 (0.71) DGAT1PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975871-B2 Continuous arycyclic compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2018-05-22 US disclosed