SCHEMBL20169425

SCHEMBL20169425

Cc1noc(-c2cc(F)ccc2C(=O)C(C)C)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.44
HCRTR1 O43613 11/20 0.42
HCRTR2 O43614 9/20 0.42
KMT2A Q03164 1/20 0.41
OPRK1 P41145 2/20 0.39
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
TACR3 P29371 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18594641 0.90 HCRTR1 (0.42) DPP4HCRTR1HCRTR2KMT2AOPRK1
SCHEMBL16114532 0.86 KMT2A (0.48) DPP4HCRTR1HCRTR2KMT2AHDAC3
SCHEMBL17071974 0.85 HCRTR1 (0.44) DPP4HCRTR1HCRTR2KMT2AOPRK1
SCHEMBL17069775 0.83 HCRTR1 (0.47) DPP4HCRTR1HCRTR2KMT2AHDAC3
SCHEMBL20169441 0.79 HCRTR1 (0.40) DPP4HCRTR1HCRTR2OPRK1
SCHEMBL17071987 0.77 KMT2A (0.44) DPP4HCRTR1HCRTR2KMT2AHDAC3
SCHEMBL10094748 0.75 NPC1 (0.44) DPP4KMT2AOPRK1
SCHEMBL18594655 0.74 HCRTR1 (0.52) HCRTR1HCRTR2KMT2AOPRK1HDAC6
SCHEMBL18163364 0.74 HCRTR1 (0.42) DPP4HCRTR1HCRTR2KMT2AOPRK1
SCHEMBL17069773 0.74 HDAC4 (0.42) HCRTR1HCRTR2KMT2AHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975876-B2 2-pyridyloxy-3-ester-4-ether orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2018-05-22 US disclosed