SCHEMBL20169441

SCHEMBL20169441

Cc1nc(-c2cc(F)ccc2C(=O)C(C)C)no1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.40
HCRTR2 O43614 3/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
BDKRB1 P46663 2/20 0.38
DPP4 P27487 2/20 0.38
DPP7 Q9UHL4 2/20 0.38
PLK1 P53350 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
OPRK1 P41145 3/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20911215 0.85 NPC1 (0.48) HCRTR1HCRTR2TRPM8PLK1L3MBTL1
SCHEMBL18594642 0.85 HCRTR1 (0.42) HCRTR1HCRTR2TRPM8PLK1L3MBTL1
SCHEMBL17069771 0.83 HCRTR1 (0.41) HCRTR1HCRTR2TRPM8PLK1L3MBTL1
SCHEMBL17071983 0.82 HCRTR1 (0.40) HCRTR1HCRTR2TRPM8PLK1L3MBTL1
SCHEMBL18594659 0.81 RAB9A (0.46) HCRTR1HCRTR2PLK1L3MBTL1LMNA
SCHEMBL20169425 0.79 DPP4 (0.44) HCRTR1HCRTR2DPP4OPRK1
SCHEMBL17071972 0.77 HCRTR1 (0.42) HCRTR1HCRTR2TRPM8PLK1L3MBTL1
SCHEMBL17723708 0.77 NPC1 (0.48) HCRTR1HCRTR2TRPM8PLK1L3MBTL1
SCHEMBL20169442 0.76 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL20928592 0.76 L3MBTL1 (0.42) TRPM8L3MBTL1OPRK1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975876-B2 2-pyridyloxy-3-ester-4-ether orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2018-05-22 US disclosed