SCHEMBL20169433

SCHEMBL20169433

CN(Cc1ccc2c(c1)C[C@H](CO[Si](C)(C)C(C)(C)C)C2)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GLS O94925 2/20 0.39
MCHR1 Q99705 5/20 0.37
HTR2C P28335 7/20 0.36
SLC6A4 P31645 7/20 0.36
HTR2A P28223 1/20 0.35
CACNA1B Q00975 2/20 0.33
CACNA1G O43497 1/20 0.33
CACNA1C Q13936 1/20 0.33
FKBP1A P62942 1/20 0.33
TOP2A P11388 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19236010 0.83 MCHR1 (0.39) GLSMCHR1HTR2CSLC6A4HTR2A
SCHEMBL17539139 0.82 GLS (0.37) GLSMCHR1HTR2CSLC6A4HTR2A
SCHEMBL17539112 0.82 GLS (0.39) GLSMCHR1HTR2CSLC6A4HTR2A
SCHEMBL17539107 0.81 GLS (0.37) GLSMCHR1HTR2CSLC6A4HTR2A
SCHEMBL17539168 0.81 GLS (0.39) GLSMCHR1HTR2CSLC6A4HTR2A
SCHEMBL17539131 0.81 GLS (0.37) GLSMCHR1HTR2CSLC6A4HTR2A
SCHEMBL17539109 0.77 GLS (0.37) GLSHTR2CSLC6A4
SCHEMBL17539104 0.77 GLS (0.36) GLSHTR2CSLC6A4
SCHEMBL20169461 0.77 GLS (0.37) GLSHTR2CSLC6A4
SCHEMBL20169457 0.77 GLS (0.36) GLSHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975848-B2 Inhibitors of HIV-1 entry and methods of use thereof THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2018-05-22 US disclosed