SCHEMBL20169442

SCHEMBL20169442

CC(C)C(=O)c1ccc(F)cc1-c1ncccn1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.46
HCRTR2 O43614 11/20 0.46
CASP6 P55212 1/20 0.40
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18594669 0.88 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL15836282 0.83 HCRTR1 (0.49) HCRTR1HCRTR2CASP6KDM4E
SCHEMBL1586269 0.81 NAPRT (0.49) HCRTR1HCRTR2CASP6KDM4E
SCHEMBL16148475 0.81 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL17069782 0.80 HCRTR1 (0.47) HCRTR1HCRTR2
SCHEMBL16025411 0.80 HCRTR1 (0.46) HCRTR1HCRTR2CASP6KDM4E
SCHEMBL19287257 0.79 PDK2 (0.42) HCRTR1HCRTR2KDM4E
SCHEMBL18163368 0.79 HCRTR1 (0.46) HCRTR1HCRTR2CASP6KDM4E
SCHEMBL20169441 0.76 HCRTR1 (0.40) HCRTR1HCRTR2
SCHEMBL19484901 0.74 HCRTR1 (0.56) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9975876-B2 2-pyridyloxy-3-ester-4-ether orexin receptor antagonists MERCK SHARP & DOHME CORP. (US) 2018-05-22 US disclosed