SCHEMBL20169979

SCHEMBL20169979

CC(C)(C)OC(=O)N1CCc2cc(C(=O)Nc3cn(I)cn3)cnc2C1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.43
MAP3K5 Q99683 7/20 0.42
NR1H2 P55055 1/20 0.42
MAPT P10636 2/20 0.41
GRAMD1A Q96CP6 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
SLC34A1 Q06495 2/20 0.37
MAPK1 P28482 1/20 0.36
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
RAF1 P04049 1/20 0.35
BRAF P15056 1/20 0.35
HPGDS O60760 1/20 0.34
GCK P35557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20364366 0.90 MAPT (0.41) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL20364368 0.87 MAP3K5 (0.40) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL20162154 0.84 MAP3K5 (0.37) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL20364367 0.82 ESR2 (0.41) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL721062 0.82 ESR2 (0.48) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL20364335 0.82 MAP3K5 (0.38) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL20364365 0.82 MAP3K5 (0.36) ESR2MAP3K5NR1H2MAPTGRAMD1A
SCHEMBL20364348 0.80 MAP3K5 (0.41) ESR2MAP3K5GCK
SCHEMBL20364356 0.80 MAP3K5 (0.41) ESR2MAP3K5MAPK1
SCHEMBL722429 0.79 ESR2 (0.49) ESR2NR1H2MAPTGRAMD1ADDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323809-A1 BICYCLIC HETEROCYCLIC AMIDE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2018-05-23 EP disclosed