SCHEMBL20169995

SCHEMBL20169995

CCc1ccc(Cl)c(C2CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 5/20 0.38
GPR84 Q9NQS5 1/20 0.38
SLC6A2 P23975 5/20 0.37
SLC6A4 P31645 5/20 0.37
SLC6A3 Q01959 5/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
TRPA1 O75762 1/20 0.36
HTR6 P50406 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35
SIGMAR1 Q99720 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15599253 0.93 SIGMAR1 (0.37) OPRL1GPR84SLC6A2SLC6A4SLC6A3
SCHEMBL20103409 0.89 ESR1 (0.39) OPRL1GPR84SLC6A2SLC6A4SLC6A3
SCHEMBL20975790 0.85 OPRL1 (0.39) OPRL1SLC6A2SLC6A4SLC6A3MEN1
SCHEMBL16962250 0.81 SLC6A2 (0.49) OPRL1GPR84SLC6A2SLC6A4SLC6A3
SCHEMBL11831337 0.78 OPRL1 (0.35) OPRL1SLC6A2SLC6A4SLC6A3MEN1
SCHEMBL18295013 0.77 SOS1 (0.40) OPRL1SLC6A2SLC6A4SLC6A3TRPA1
SCHEMBL10829892 0.77 SIGMAR1 (0.48) HTR6SIGMAR1
SCHEMBL11835240 0.75 OPRL1 (0.39) OPRL1SLC6A2SLC6A4SLC6A3SIGMAR1
SCHEMBL16961163 0.74 OPRL1 (0.39) OPRL1SLC6A2SLC6A4SLC6A3TRPA1
SCHEMBL20889624 0.74 CYP2A6 (0.42) OPRL1MEN1KMT2ATRPA1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323809-A1 BICYCLIC HETEROCYCLIC AMIDE DERIVATIVE Sumitomo Dainippon Pharma Co., Ltd. (JP) 2018-05-23 EP disclosed