SCHEMBL20170488

SCHEMBL20170488

CC(=O)Nc1ncc(S(=O)(=O)N2Cc3cccc(-c4cncn4F)c3C2)s1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.37
LPAR1 Q92633 1/20 0.36
LPAR2 Q9HBW0 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 2/20 0.34
OGA O60502 3/20 0.33
LIMK1 P53667 1/20 0.33
POLB P06746 1/20 0.32
IDO1 P14902 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
S1PR1 P21453 1/20 0.31
PIK3CG P48736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719059 0.83 MGAT2 (0.34) SCN9ALPAR1LPAR2SMN1; SMN2PKM
SCHEMBL16730885 0.78 SCN9A (0.38) SCN9ALPAR1LPAR2SMN1; SMN2LMNA
SCHEMBL20170497 0.78 SCN9A (0.38) SCN9ALPAR1LPAR2SMN1; SMN2LMNA
SCHEMBL16730892 0.77 OGA (0.35) SCN9ALPAR1LPAR2SMN1; SMN2PKM
SCHEMBL1000263 0.71 LPAR1 (0.51) SCN9ALPAR1LPAR2LMNAOGA
SCHEMBL16903932 0.68 POLB (0.53) SCN9ALPAR1LPAR2SMN1; SMN2LMNA
SCHEMBL1058013 0.66 L3MBTL1 (0.52) SCN9ALPAR1LPAR2SMN1; SMN2RAB9A
SCHEMBL16720931 0.65 OGA (0.36) SCN9ALPAR1LPAR2OGA
SCHEMBL16718968 0.65 DRD3 (0.35) SCN9AIDO1MEN1KMT2A
SCHEMBL16718995 0.65 OGA (0.38) SMN1; SMN2LMNAOGAIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed