SCHEMBL20170511

SCHEMBL20170511

CC(c1ccc(F)cc1)n1cncc1-c1cccc2c1CCN(S(=O)(=O)c1cnc(N)s1)C2

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 12/20 0.36
SIGMAR1 Q99720 3/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
KCNK3 O14649 3/20 0.33
SCN5A Q14524 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16730893 1.00 SCN9A (0.36) SCN9ASIGMAR1MEN1KMT2AKCNK3
SCHEMBL16730881 0.92 SCN9A (0.36) SCN9ASIGMAR1MEN1KMT2AKCNK3
SCHEMBL20170497 0.87 SCN9A (0.38) SCN9ASCN5A
SCHEMBL16730885 0.87 SCN9A (0.38) SCN9ASCN5A
SCHEMBL18128784 0.83 KCNK3 (0.35) SIGMAR1MEN1KMT2AKCNK3
SCHEMBL16731014 0.83 KCNK3 (0.35) SIGMAR1MEN1KMT2AKCNK3
SCHEMBL20170445 0.82 PRCP (0.35) SCN9AMEN1KMT2A
SCHEMBL16718972 0.81 SCN9A (0.31) SCN9A
SCHEMBL20162455 0.81 SCN9A (0.31) SCN9A
SCHEMBL16903905 0.77 POLB (0.40) SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068391-B1 ARYL LINKED IMIDAZOLE AND TRIAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR IMPROVING THE PHARMACOKINETICS OF A DRUG MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed