SCHEMBL20170552

SCHEMBL20170552

CC(O)C(NC(=O)NCc1nnc(C(N)C(C)O)o1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 6/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
CD274 Q9NZQ7 4/20 0.40
VSIR Q9H7M9 3/20 0.40
PDCD1LG2 Q9BQ51 2/20 0.39
MAPK1 P28482 1/20 0.36
TSHR P16473 1/20 0.36
PDCD1 Q15116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19413592 0.91 HDAC8 (0.42) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170542 0.91 HDAC8 (0.42) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170558 0.88 CD274 (0.50) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170520 0.88 CD274 (0.50) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170571 0.87 CD274 (0.49) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170572 0.87 CD274 (0.49) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL19969086 0.87 CD274 (0.44) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170534 0.86 HDAC8 (0.42) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170543 0.86 HDAC8 (0.42) HDAC8HDAC1HDAC2CD274VSIR
SCHEMBL20170561 0.85 CD274 (0.41) HDAC8HDAC1HDAC2CD274VSIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041828-B1 1,3,4-OXADIAZOLE AND 1,3,4-THIADIAZOLE DERIVATIVES AS IMMUNOMODULATORS AURIGENE DISCOVERY TECH LTD (IN) 2018-05-23 EP disclosed