SCHEMBL20170674

SCHEMBL20170674

CCN(C)[C@H]1Cc2ccc(OC)c3c2C2C1CC[C@H](O)[C@H]2O3

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.51
OPRM1 P35372 9/20 0.43
OPRK1 P41145 3/20 0.37
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13014030 1.00 HCRTR1 (0.51) HCRTR1OPRM1OPRK1HTR1A
SCHEMBL18473573 0.88 HCRTR1 (0.49) HCRTR1OPRM1OPRK1
SCHEMBL13079206 0.79 OPRM1 (0.43) HCRTR1OPRM1OPRK1
SCHEMBL10223933 0.76 HCRTR1 (0.45) HCRTR1OPRM1OPRK1HTR1A
SCHEMBL18473435 0.73 HCRTR1 (0.42) HCRTR1OPRM1HTR1A
SCHEMBL20170652 0.72 OPRM1 (0.37) HCRTR1OPRM1
SCHEMBL20170728 0.72 OPRM1 (0.37) HCRTR1OPRM1
SCHEMBL20170607 0.72 OPRM1 (0.37) HCRTR1OPRM1
SCHEMBL20170820 0.71 HCRTR1 (0.46) HCRTR1OPRM1OPRK1
SCHEMBL13072118 0.70 OPRM1 (0.50) HCRTR1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2453895-B1 (+) - MORPHINANS AS ANTAGONISTS OF TOLL-LIKE RECEPTOR 9 AND THERAPEUTIC USES THEREOF MALLINCKRODT LLC (US) 2018-05-23 EP disclosed