SCHEMBL20171265

SCHEMBL20171265

NC(=O)c1ncc(-c2cncnc2)cc1O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.43
EGLN1 Q9GZT9 10/20 0.39
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
ERN1 O75460 1/20 0.39
FLT1 P17948 4/20 0.39
VEGFA P15692 3/20 0.39
MKNK1 Q9BUB5 4/20 0.39
MKNK2 Q9HBH9 4/20 0.39
LRRK2 Q5S007 1/20 0.39
AR P10275 1/20 0.37
EGLN3 Q9H6Z9 4/20 0.37
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24405092 0.83 EGLN1 (0.40) CYP11B2EGLN1ERN1FLT1VEGFA
SCHEMBL22462719 0.77 EGLN1 (0.60) EGLN1IKBKBFLT1VEGFAMKNK1
SCHEMBL28778074 0.76 EGLN1 (0.43) EGLN1FLT1VEGFAEGLN3
SCHEMBL28778073 0.75 GSK3B (0.40) CYP11B2IKBKBCHUKERN1MKNK1
SCHEMBL14152807 0.74 EGLN1 (0.62) EGLN1FLT1VEGFALRRK2EGLN3
SCHEMBL1923191 0.74 EGLN1 (0.73) EGLN1FLT1VEGFAEGLN3
SCHEMBL1055362 0.74 SPR (0.44) CHUKMKNK1MKNK2
SCHEMBL27772404 0.74 KMT2A (0.38) EGLN1FLT1VEGFA
SCHEMBL15641357 0.73 EGLN1 (0.61) EGLN1FLT1VEGFALRRK2EGLN3
SCHEMBL3031409 0.73 EGLN1 (0.63) EGLN1IKBKBFLT1VEGFAEGLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3357911-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE Akebia Therapeutics Inc. (US) 2018-08-08 EP disclosed
EP-3323807-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE Akebia Therapeutics, Inc. (US) 2018-05-23 EP disclosed