SCHEMBL20171906

SCHEMBL20171906

CC(C)(C)COc1nc(N2CCOCC2)c2nc[nH]c2n1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.44
LRRK2 Q5S007 3/20 0.38
CHEK1 O14757 4/20 0.38
MAPK1 P28482 2/20 0.38
PDPK1 O15530 1/20 0.38
PAK1 Q13153 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
JAK2 O60674 1/20 0.35
ZAP70 P43403 1/20 0.35
SYK P43405 1/20 0.35
PIK3CA P42336 2/20 0.35
MTOR P42345 2/20 0.35
PIK3CG P48736 2/20 0.35
RAF1 P04049 1/20 0.35
BRAF P15056 1/20 0.35
JAK3 P52333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16211956 0.83 CNR2 (0.52) CNR2
SCHEMBL16211738 0.80 CNR2 (0.70) CNR2
SCHEMBL16211686 0.79 CNR2 (0.54) CNR2
SCHEMBL16222478 0.79 CNR2 (0.58) CNR2
SCHEMBL20171935 0.78 MAPK1 (0.43) LRRK2CHEK1MAPK1PDPK1PAK1
SCHEMBL14071958 0.77 MAP2K7 (0.45) LRRK2CHEK1MAPK1PDPK1PAK1
SCHEMBL8826341 0.74 IKBKB (0.52) LRRK2CHEK1MAPK1PDPK1PAK1
SCHEMBL30253959 0.74 CHEK1 (0.44) LRRK2CHEK1MAPK1PDPK1PAK1
SCHEMBL336113 0.74 CHEK1 (0.44) LRRK2CHEK1MAPK1PDPK1PAK1
SCHEMBL19414424 0.74 CHEK1 (0.44) CHEK1MAPK1PDPK1PAK1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991987-B1 PURINE DERIVATIVES AS CB2 RECEPTOR AGONISTS HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed