SCHEMBL20171945

SCHEMBL20171945

ClC1=NCCc2occc21

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.36
HSD17B10 Q99714 3/20 0.34
POLB P06746 2/20 0.34
GAA P10253 1/20 0.34
KDM4E B2RXH2 2/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP19A1 P11511 2/20 0.31
TBXAS1 P24557 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18903799 0.71 MAPK10 (0.40) HSP90AA1HSD17B10POLBGAAKDM4E
SCHEMBL18903831 0.66 NISCH (0.34) POLBMAPT
SCHEMBL15037590 0.66 HSP90AA1 (0.33) HSP90AA1CYP19A1TBXAS1
SCHEMBL449725 0.61
SCHEMBL21025349 0.60 PARP10 (0.46) KDM4E
SCHEMBL583280 0.58
SCHEMBL3129135 0.58 HSD17B10 (0.39) HSP90AA1HSD17B10POLBGAAKDM4E
SCHEMBL15395750 0.58 HSP90AA1 (0.38) HSP90AA1HSD17B10POLBGAAKDM4E
SCHEMBL13090140 0.58 MAPT (0.39) HSP90AA1HSD17B10POLBGAAKDM4E
SCHEMBL333300 0.58 MAPT (0.42) HSP90AA1HSD17B10POLBGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323821-A1 HETEROAROMATIC COMPOUNDS AND THEIR USE AS DOPAMINE D1 LIGANDS Pfizer Inc (US) 2018-05-23 EP disclosed