SCHEMBL20172385

SCHEMBL20172385

CCc1ccc2c(ccn2Cc2cccc(F)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 10/20 0.53
PPARG P37231 9/20 0.53
MAOB P27338 1/20 0.48
SLC2A1 P11166 1/20 0.48
EGFR P00533 2/20 0.47
PLAU P00749 2/20 0.47
PLG P00747 1/20 0.47
ERBB2 P04626 1/20 0.45
DBH P09172 1/20 0.45
DPP4 P27487 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
PDE1A P54750 1/20 0.42
PDE1B Q01064 1/20 0.42
PDE1C Q14123 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11949599 0.84 DPP4 (0.53) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL16783105 0.84 APP (0.52) PLAUPLGERBB2
SCHEMBL3507375 0.82 EGFR (0.62) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL6085951 0.82 EGFR (0.51) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL15701546 0.81 KCNH2 (0.49) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL31258087 0.81 HTR6 (0.55) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL1104768 0.81 HTR6 (0.55) EPHX2PPARGMAOBSLC2A1EGFR
Ethoxycarbonyl Group SCHEMBL28763762 0.79 EPHX2 (0.47) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL4194376 0.76 IDO1 (0.54) EPHX2PPARGMAOBSLC2A1EGFR
SCHEMBL9584191 0.76 APP (0.53) PPARGPLAUPLGERBB2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2680850-B1 ALKYNE SUBSTITUTED QUINAZOLINE COMPOUND AND METHODS OF USE NEWGEN THERAPEUTICS INC (US) 2018-05-23 EP disclosed