SCHEMBL20172422

SCHEMBL20172422

Cc1ccc(Oc2ccn3ncnc3c2)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 11/20 0.40
EGFR P00533 8/20 0.40
NQO2 P16083 1/20 0.40
FECH P22830 1/20 0.40
MYH14 Q7Z406 1/20 0.40
RIPK3 Q9Y572 1/20 0.40
ERBB3 P21860 1/20 0.38
ERBB4 Q15303 1/20 0.38
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13655122 0.86 ERBB2 (0.47) ERBB2EGFRNQO2FECHMYH14
SCHEMBL3484112 0.84 EGFR (0.38) ERBB2EGFRNQO2FECHMYH14
SCHEMBL29887886 0.84 EGFR (0.38) ERBB2EGFRNQO2FECHMYH14
SCHEMBL15703717 0.84 CYP2C19 (0.40) ERBB2EGFRNQO2FECHMYH14
SCHEMBL12524904 0.82 SCN5A (0.39) ERBB2EGFRERBB3ERBB4MEN1
SCHEMBL26580265 0.81 ERBB2 (0.42) ERBB2EGFRNQO2FECHMYH14
SCHEMBL18181595 0.80 TEAD4 (0.38) ERBB2EGFRNQO2FECHMYH14
SCHEMBL24569945 0.79 PDE7A (0.52) MEN1KMT2A
SCHEMBL29834731 0.79 PDE7A (0.52) MEN1KMT2A
SCHEMBL26894024 0.78 ERBB2 (0.43) ERBB2EGFRNQO2FECHMYH14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2680850-B1 ALKYNE SUBSTITUTED QUINAZOLINE COMPOUND AND METHODS OF USE NEWGEN THERAPEUTICS INC (US) 2018-05-23 EP disclosed