SCHEMBL20172635

SCHEMBL20172635

N#CCNC(=O)[C@@H]1CNCCCO1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 19/20 0.47
KCNH2 Q12809 2/20 0.47
SSTR4 P31391 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26081106 1.00 CTSC (0.47) CTSCKCNH2SSTR4
SCHEMBL25046589 0.78 SSTR4 (0.49) CTSCKCNH2SSTR4
SCHEMBL24973027 0.77 CTSC (0.54) CTSCKCNH2
SCHEMBL6039537 0.77 SSTR4 (0.49) CTSCSSTR4
Hydrochloric Acid SCHEMBL29189762 0.76 SSTR4 (0.48) CTSCKCNH2SSTR4
SCHEMBL26668539 0.76 SSTR4 (0.48) CTSCSSTR4
SCHEMBL24697125 0.75 CTSK (0.43)
SCHEMBL24697974 0.75 CTSK (0.43)
SCHEMBL8860932 0.74 SSTR4 (0.52) CTSCSSTR4
SCHEMBL18664465 0.74 SSTR4 (0.52) CTSCSSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4129989-A1 NITRILE DERIVATIVE THAT ACTS AS INHIBITOR OF DIPEPTIDYL PEPTIDASE 1 AND USE THEREOF Haisco Pharmaceuticals Pte. Ltd. (SG) 2023-02-08 EP disclosed
EP-3323814-B1 (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2020-05-13 EP disclosed
EP-3323814-A1 (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES AS DIPEPTIDYL PEPTIDASE I INHIBITORS AstraZeneca AB (SE) 2018-05-23 EP disclosed