SCHEMBL20174403

SCHEMBL20174403

c1ccc(-c2ccc(-c3ccc4c(c3)C3(c5ccccc5-c5ccccc53)c3oc5ccccc5c3-4)cc2)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 8/20 0.43
DHODH Q02127 1/20 0.33
HSD11B1 P28845 1/20 0.33
NPY5R Q15761 1/20 0.32
HSD17B10 Q99714 2/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ALK Q9UM73 1/20 0.31
AHR P35869 1/20 0.31
PRKDC P78527 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20174423 0.93 PDK2 (0.40) PDK2DHODHHSD11B1NPY5RHSD17B10
SCHEMBL20174416 0.89 PDK2 (0.44) PDK2DHODHHSD11B1NPY5RHSD17B10
SCHEMBL20174419 0.87 PDK2 (0.46) PDK2ALK
SCHEMBL20174398 0.84 PDK2 (0.39) PDK2DHODHMAPK1
SCHEMBL20174361 0.84 PDK2 (0.39) PDK2DHODHMAPK1
SCHEMBL20174322 0.84 PDK2 (0.39) PDK2DHODHMAPK1
SCHEMBL20174441 0.84 KDM4E (0.34) PDK2HSD17B10TSHRKDM4EALDH1A1
SCHEMBL20199301 0.84 PDK2 (0.45) PDK2MAPK1ALDH1A1AHR
SCHEMBL20174393 0.83 KMT2A (0.37) PDK2DHODHMAPK1KDM4EALDH1A1
SCHEMBL19008461 0.83 KMT2A (0.37) PDK2DHODHMAPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10738034-B2 Spiro compound and organic light-emitting device comprising same LG CHEM, LTD. (KR) 2020-08-11 US disclosed
US-20180141933-A1 SPIRO COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME LG CHEM, LTD. (KR) 2018-05-24 US disclosed
US-20180141933-A1 SPIRO COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME LG CHEM, LTD. (KR) 2018-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10738034-B2 Spiro compound and organic light-emitting device comprising same CRY1, NR2E3, ERG PDK2 651/4885DHODH 189/4885HSD11B1 196/4885
US-20180141933-A1 SPIRO COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME CRY1, NR2E3, ERG PDK2 651/4885DHODH 189/4885HSD11B1 196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.