SCHEMBL20176607

SCHEMBL20176607

COc1ccc(Cn2ncc3c(Br)cc(I)cc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 5/20 0.49
PDE1B Q01064 5/20 0.49
PDE1C Q14123 5/20 0.49
NPBWR1 P48145 8/20 0.45
PKM P14618 1/20 0.45
PKLR P30613 1/20 0.45
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42
MCHR1 Q99705 1/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B3 P37058 1/20 0.40
BRD4 O60885 1/20 0.40
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22139429 0.80 NPBWR1 (0.48) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL22913090 0.80 NPBWR1 (0.51) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL22912921 0.80 PDE1B (0.49) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL21608784 0.77 NPBWR1 (0.45) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL2443709 0.76 NPBWR1 (0.47) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL29514413 0.76 PDE1B (0.50) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL29049927 0.76 PDE1B (0.50) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL16014472 0.75 PDE1A (0.50) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL18428510 0.74 PDE1A (0.49) PDE1APDE1BPDE1CNPBWR1PKM
SCHEMBL27077682 0.74 NPBWR1 (0.57) PDE1APDE1BPDE1CNPBWR1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092047-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE JOINT STOCK COMPANY "BIOCAD" (RU) 2018-05-24 WO disclosed