SCHEMBL2017789

SCHEMBL2017789

N#Cc1ccc(N2CCC(C(=O)N3CC[C@H](c4ccc(Cl)cc4)C3)CC2)nn1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 15/20 0.57
PANK3 Q9H999 4/20 0.52
RIPK1 Q13546 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12517729 0.84 TACR3 (0.61) TACR3PANK3
SCHEMBL2017867 0.84 PANK3 (0.57) TACR3PANK3RIPK1
SCHEMBL15751845 0.80 TACR3 (0.67) TACR3
SCHEMBL6903622 0.79 TACR3 (0.63) TACR3
SCHEMBL15751844 0.79 TACR3 (0.58) TACR3RIPK1
SCHEMBL1439412 0.75 TACR3 (0.57) TACR3
SCHEMBL12789428 0.75 TACR3 (0.61) TACR3
SCHEMBL1439342 0.75 TACR3 (0.61) TACR3
SCHEMBL1439340 0.75 TACR3 (0.61) TACR3
SCHEMBL1978749 0.74 TACR3 (0.84) TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO claimed
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed