SCHEMBL2017867

SCHEMBL2017867

N#Cc1ccc(N2CCC(c3ccc(Cl)cc3)CC2)nn1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PANK3 Q9H999 10/20 0.57
TACR3 P29371 4/20 0.46
RIPK1 Q13546 1/20 0.43
GRM2 Q14416 1/20 0.43
RET P07949 1/20 0.42
DRD2 P14416 1/20 0.41
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
JAK3 P52333 1/20 0.39
SLC18A3 Q16572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2017789 0.84 TACR3 (0.57) PANK3TACR3RIPK1
SCHEMBL2016712 0.80 RET (0.48) PANK3TACR3RIPK1GRM2RET
SCHEMBL17687600 0.77 PANK3 (0.48) PANK3RIPK1JAK2JAK1JAK3
SCHEMBL24536328 0.74 PANK3 (0.49) PANK3RIPK1JAK2JAK1JAK3
SCHEMBL12683340 0.74 CYP1A2 (0.52) PANK3RIPK1
SCHEMBL19748509 0.73 PANK3 (1.00) PANK3
SCHEMBL21424030 0.73 PANK3 (0.64) PANK3
SCHEMBL23750439 0.73 PANK3 (0.70) PANK3
Hydrochloric Acid SCHEMBL17687632 0.72 JAK2 (0.47) PANK3RIPK1JAK2JAK1JAK3
SCHEMBL24536005 0.71 PANK3 (0.47) PANK3RIPK1JAK2JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513084-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed