SCHEMBL20180069

SCHEMBL20180069

COC(=O)CN(CCN(CCN(CC(=O)O)CC(=O)O)Cc1ccc(C=O)cc1)CC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 13/20 0.41
CA2 P00918 13/20 0.41
CA4 P22748 6/20 0.41
ALDH1A1 P00352 1/20 0.39
NR1D1 P20393 1/20 0.38
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
EYA2 O00167 1/20 0.37
APP P05067 1/20 0.37
ACE P12821 1/20 0.37
CA12 O43570 2/20 0.36
CA9 Q16790 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRA2A P08913 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
DRD1 P21728 1/20 0.36
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22147372 0.89 TDP1 (0.47) CA1CA2CA4ALDH1A1KMT2A
SCHEMBL14341631 0.82 NR1D1 (0.40) CA1CA2CA4NR1D1
SCHEMBL12198408 0.78 NPC1 (0.47) ALDH1A1KMT2ATDP1CA12CA9
SCHEMBL10958880 0.78 NR1D1 (0.51) ALDH1A1NR1D1KMT2AKDM4ELMNA
Edetic Acid SCHEMBL3810362 0.76 TDP1 (0.64) CA1CA2CA4KMT2ATDP1
SCHEMBL5852235 0.76 TDP1 (0.64) CA1CA2CA4KMT2ATDP1
SCHEMBL5852270 0.76 TDP1 (0.64) CA1CA2CA4KMT2ATDP1
SCHEMBL13129733 0.76 TDP1 (0.64) CA1CA2CA4KMT2ATDP1
SCHEMBL5085940 0.76 TDP1 (0.64) CA1CA2CA4KMT2ATDP1
SCHEMBL14355755 0.76 NR1D1 (0.43) ALDH1A1NR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541368-B1 IMAGEABLE PARTICLES, METHODS OF MAKING AND METHODS OF USE THEREOF US HEALTH (US) 2023-07-12 EP disclosed
WO-2018093566-A1 IMAGEABLE PARTICLES, METHODS OF MAKING AND METHODS OF USE THEREOF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2018-05-24 WO disclosed