SCHEMBL20180748

SCHEMBL20180748

C[C@@H]1CN(c2ccc(N)cc2Cl)C[C@H](C)N1C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.62
HTT P42858 1/20 0.62
MAPT P10636 6/20 0.59
KDM4E B2RXH2 1/20 0.59
RAD52 P43351 1/20 0.59
POLB P06746 2/20 0.56
GAA P10253 4/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
TDP1 Q9NUW8 1/20 0.43
CYP3A4 P08684 3/20 0.43
NFKB1 P19838 1/20 0.40
PMP22 Q01453 1/20 0.40
MEN1 O00255 1/20 0.39
THRB P10828 1/20 0.39
NR4A1 P22736 1/20 0.39
KMT2A Q03164 1/20 0.39
PTK2B Q14289 1/20 0.39
TSHR P16473 1/20 0.38
RECQL P46063 1/20 0.38
HTR1D P28221 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20180601 0.82 ALDH1A1 (0.41) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL29533302 0.82 MAPT (0.56) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL23262628 0.82 MAPT (0.56) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL11202420 0.82 ALDH1A1 (0.69) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL10126811 0.82 MAPT (0.56) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL1046324 0.81 ALDH1A1 (0.49) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL29532627 0.81 ALDH1A1 (0.40) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL23246126 0.81 ALDH1A1 (0.40) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL14320572 0.81 ALDH1A1 (0.62) ALDH1A1HTTMAPTKDM4ERAD52
SCHEMBL1046325 0.81 ALDH1A1 (0.49) ALDH1A1HTTMAPTKDM4ERAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019011228-A1 IMIDAZO[1,2-B]PYRIMIDO[4,5-D]PYRIDAZIN-5(6H)-ONE COMPOUND AND USE THEREOF 上海瑛派药业有限公司 2019-01-17 WO disclosed
WO-2018090939-A1 8,9-DIHYDROIMIDAZOLE[1,2-A]PYRIMIDO[5,4-E]PYRIMIDINE-5(6H)-KETONE COMPOUND 上海瑛派药业有限公司 2018-05-24 WO disclosed