SCHEMBL20182200

SCHEMBL20182200

CC(/C(=C/Nc1ccccc1F)N=N)n1cc(-c2ccc(OC3CC3)nc2)c2c(N)ncnc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.39
TEK Q02763 9/20 0.39
LCK P06239 6/20 0.39
SRC P12931 3/20 0.39
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
PRKDC P78527 1/20 0.36
HCK P08631 3/20 0.35
FLT3 P36888 2/20 0.35
NEK7 Q8TDX7 2/20 0.35
KCNH2 Q12809 1/20 0.34
BTK Q06187 1/20 0.34
EIF2AK3 Q9NZJ5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182298 0.93 NEK7 (0.38) KDRTEKLCKSRCPIK3CD
SCHEMBL20182228 0.91 KDR (0.45) KDRTEKLCKSRCHCK
SCHEMBL20182362 0.86 CFTR (0.40) KDRTEKLCKSRCPIK3CD
SCHEMBL20181890 0.83 KDR (0.44) KDRTEKLCKSRCPIK3CD
SCHEMBL20182204 0.81 KDR (0.37) KDRTEKLCKSRCPIK3CD
SCHEMBL20182241 0.81 KDR (0.46) KDRTEKLCKSRCPIK3CD
SCHEMBL20181904 0.81 PDPK1 (0.36) KDRTEKLCKSRCPIK3CD
SCHEMBL20181907 0.79 EGFR (0.35) KDRTEKLCKSRC
SCHEMBL20182274 0.78 EIF2AK3 (0.40) KDRTEKLCKSRCPIK3CD
SCHEMBL20181883 0.78 NTRK1 (0.40) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed